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奈妥吡坦 Netupitant

奈妥吡坦 Netupitant

【化學(xué)名】奈妥吡坦 Netupitant

【原研】羅氏

【上市時間】20141010

【用途】用于治療惡心,嘔吐

【劑型/規(guī)格】膠囊 300mg;EQ 0.5mg BASE ;凍干 EQ 235MG BASE/VIAL;EQ 0.25MG BASE/VIAL ;靜脈注射液 EQ 235MG BASE/20ML (EQ 11.75MG BASE/ML);EQ 0.25MG BASE/20ML (EQ 0.0125MG BASE/ML)



奈妥吡坦Netupitant

 

一、產(chǎn)品概述

Netupitant奈妥匹坦,由羅氏首先研發(fā),用于治療惡心、嘔吐;后由Helsinn研發(fā)其復(fù)方制劑奈妥吡坦/鹽酸帕洛諾司瓊。2014年10月10日,奈妥吡坦/鹽酸帕洛諾司瓊獲得FDA批準,由赫爾辛醫(yī)療股份公司銷售,商品名為Akynzeo

 

二、主要產(chǎn)品

Description

Structural Formula

CAS No.

Category

Netupitant

API.png

290297-26-6

API

2-(3,5-bis(trifluoromethyl)   phenyl)-2-methylpropanoic acid

70-0.png

289686-70-0

intermediates

3-Pyridinecarboxamide,

4-(2-methylphenyl)-6-(4-methyl-1-piperazinyl)-  

01-0.png

342417-01-0

intermediates

3-Pyridinamine,N-methyl-4-(2-methylphenyl)-6-(4-methyl-1-piperazinyl)-

25-5.png


290297-25-5

intermediates

Note: Products protected by valid patents are not offered for sale in countries where the sale of such products constitutes patent infringement and its liability is at buyer's risk.

 


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