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Seladelpar lysine dihydrate MBX-8052

Seladelpar lysine dihydrate MBX-8052


【化學(xué)名】Seladelpar lysine dihydrate

【原研】Cymabay Therapeutics Inc

【上市時(shí)間】2024年08月14日

【用途】用于治療硬化性膽管炎

【劑型/規(guī)格】口服膠囊劑,規(guī)格EQ 10MG BASE


Seladelpar lysine dihydrate  MBX-8052

 

一、產(chǎn)品概述

Seladelpar lysine dihydrate是由Cymabay Therapeutics Inc研發(fā)的一種小分子藥物,是一種PPARδ激動(dòng)劑。該藥物于2024年08月14日獲FDA批準(zhǔn),用于治療硬化性膽管炎。

二、主要產(chǎn)品

Description

Structural Formula

CAS No.

Category

Seladelpar lysine dihydrate

API.png

928821-40-3

API

ethyl   2-(4-mercapto-2-methylphenoxy)acetate

82-7.png

343322-82-7

intermediates

(R)-2-((4-(trifluoromethyl)phenoxy)methyl)oxirane

58-4.png

256372-58-4

intermediates

Note: Products protected by valid patents are not offered for sale in countries where the sale of such products constitutes patent infringement and its liability is at buyer's risk.



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